Bremelanotide Muscle Building Supplements PT-141T Sexual Desire Increasing

Product Details:
Place of Origin: China
Brand Name: Filter
Certification: GMP
Model Number: 189691-06-3
Payment & Shipping Terms:
Minimum Order Quantity: 10vials
Price: Negotiable
Packaging Details: Plastic ,bubble, silver paper, 1kg/bag, 100g/bag
Delivery Time: 1-2 works day
Payment Terms: T/T, Western Union, MoneyGram
Supply Ability: 10000vial / month

Detail Information

Color: White Form: Powder
Name: PT-141 Specifications: 10mg
Other Name: Bremelanotide
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Product Description

Pharmaceutical Peptide Bremelanotide 32780-32-8 PT-141

 

CAS No.: 32780-32-8 Other Names: PT 141 MF: C7H15NO4
EINECS No.: 258279-04-8 Place of Origin: ShangHai, China (Mainland) Type: Auxiliaries and Other Medicinal Chemicals
Grade Standard: Medicine Grade Usage: Animal Pharmaceuticals, Bodybuilding    
Model Number:   Purity: 99%min Product Name: PT141
Appearance: Powder Grade: Medical Standard: USP Grade
Colour: White Export Markets: Global Production Capacity: 10000g
   


Description
PT-141 (Bremelanotide) is a highly potent synthetic peptide analogue of α-MSH that may elicit aphrodisiac effects through stimulation of melanocortin receptors. PT-141 (Bremelanotide) consists of seven amino acids and is a cyclic, shortened lactam variant of alpha-Melanocyte-stimulating hormone (α-MSH), a multifunctional peptide that regulates a broad array of physiological functions. In studies, bremelanotide was shown to induce lordosis in an animal model and was also effective in treating sexual dysfunction in both men (erectile dysfunction or impotence) and women (sexual arousal disorder).

Specification
Name: PT-141
Synonyms: Bremelanotide, PT-141 Acetate
CAS #: 189691-06-3
Molecular Formula: C50H68N14O10
Molecular Mass: 1025.2 Da (g/mol)
Amino Acid Sequence: Ac-Nle-cyclo[Asp-His-D-Phe-Arg-Trp-Lys]-OH

Purity
PT-141 has a peptide purity level that exceeds 99.0% as determined by HPLC and MS. This peptide was synthesized with no additives and is supplied as a white lyophilized (freeze-dried) powder.

Usage
Bremelanotide, similarly to its analogues α-MSH and melanotan II, acts as a non-selective agonist of all of the melanocortin receptors except MC2, where it lacks significant affinity. Reported activity of the drug is as follows:
MC1 (Ki = 0.68 nM)
MC2 (Ki > 1000 nM)
MC3 (Ki = 72.07 nM)
MC4 (Ki = 19.25 nM)
MC5 (Ki = 166.8 nM)

Bremelanotide appears to stimulate sexual desire and arousal completely or mostly via activation of the MC4 receptor (the MC3 receptor may also be involved). It modulates inflammation and limits ischemia via activation of the MC1 and MC4 receptors.

According to Palatin Technologies' original 2003 patent for bremelanotide, it possesses approximately 50 times the potency of melanotan II as an inducer of erection in male rats. In addition, it was stated in the patent that the therapeutic window of bremelanotide in animals (specifically, the range of induction of the desired sexual arousal relative to the induction of side effects including nausea, yawning, stretching, and decreased appetite) was >1,000-fold, whereas that of melanotan II was only 3- to 4-fold. They concluded that bremelanotide would be more tolerable than melanotan II.

 

Bremelanotide Muscle Building Supplements PT-141T Sexual Desire Increasing 0

Bremelanotide Muscle Building Supplements PT-141T Sexual Desire Increasing 1

-----------Additional Information ------------
Brand: Filter
Package: Plastic Tube
Place of origin: China
Certificate: GMP
Port: Shanghai,Guangzhou,Shenzhen,HongKong

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